| The dTAG system for immediate and target-specific protein degradation B Nabet, JM Roberts, DL Buckley, J Paulk, S Dastjerdi, A Yang, ... Nature chemical biology 14 (5), 431-441, 2018 | 718 | 2018 |
| Pharmacological perturbation of CDK9 using selective CDK9 inhibition or degradation CM Olson, B Jiang, MA Erb, Y Liang, ZM Doctor, Z Zhang, T Zhang, ... Nature chemical biology 14 (2), 163-170, 2018 | 430 | 2018 |
| BET bromodomain proteins function as master transcription elongation factors independent of CDK9 recruitment GE Winter, A Mayer, DL Buckley, MA Erb, JE Roderick, S Vittori, JM Reyes, ... Molecular cell 67 (1), 5-18. e19, 2017 | 391 | 2017 |
| Transcription control by the ENL YEATS domain in acute leukaemia MA Erb, TG Scott, BE Li, H Xie, J Paulk, HS Seo, A Souza, JM Roberts, ... Nature 543 (7644), 270-274, 2017 | 297 | 2017 |
| ENL links histone acetylation to oncogenic gene expression in acute myeloid leukaemia L Wan, H Wen, Y Li, J Lyu, Y Xi, T Hoshii, JK Joseph, X Wang, YHE Loh, ... Nature 543 (7644), 265-269, 2017 | 240 | 2017 |
| Functional TRIM24 degrader via conjugation of ineffectual bromodomain and VHL ligands LN Gechijian, DL Buckley, MA Lawlor, JM Reyes, J Paulk, CJ Ott, ... Nature chemical biology 14 (4), 405-412, 2018 | 213 | 2018 |
| Enhancer invasion shapes MYCN-dependent transcriptional amplification in neuroblastoma R Zeid, MA Lawlor, E Poon, JM Reyes, M Fulciniti, MA Lopez, TG Scott, ... Nature genetics 50 (4), 515-523, 2018 | 194 | 2018 |
| Translation Termination Factor GSPT1 Is a Phenotypically Relevant Off-Target of Heterobifunctional Phthalimide Degraders M Ishoey, S Chorn, N Singh, MG Jaeger, M Brand, J Paulk, S Bauer, ... ACS chemical biology 13 (3), 553-560, 2018 | 144 | 2018 |
| Chemical inhibition of ENL/AF9 YEATS domains in acute leukemia L Garnar-Wortzel, TR Bishop, S Kitamura, N Milosevich, JN Asiaban, ... ACS central science 7 (5), 815-830, 2021 | 49 | 2021 |
| A short ORF-encoded transcriptional regulator M Koh, I Ahmad, Y Ko, Y Zhang, TF Martinez, JK Diedrich, Q Chu, ... Proceedings of the National Academy of Sciences 118 (4), e2021943118, 2021 | 37 | 2021 |
| Cell-based ligand discovery for the ENL YEATS domain JN Asiaban, N Milosevich, E Chen, TR Bishop, J Wang, Y Zhang, ... ACS Chemical Biology 15 (4), 895-903, 2020 | 35 | 2020 |
| Insights into the mechanism of cell death induced by saporin delivered into cancer cells by an antibody fusion protein targeting the transferrin receptor 1 TR Daniels-Wells, G Helguera, JA Rodríguez, LS Leoh, MA Erb, ... Toxicology in Vitro 27 (1), 220-231, 2013 | 35 | 2013 |
| Pharmacological Modulation of Transcriptional Coregulators in Cancer TR Bishop, Y Zhang, MA Erb Trends in pharmacological sciences 40 (6), 388-402, 2019 | 15 | 2019 |
| Acetyl-CoA biosynthesis drives resistance to histone acetyltransferase inhibition TR Bishop, C Subramanian, EM Bilotta, L Garnar-Wortzel, AR Ramos, ... Nature Chemical Biology 19 (10), 1215-1222, 2023 | 7 | 2023 |
| Collateral lethality between HDAC1 and HDAC2 exploits cancer-specific NuRD complex vulnerabilities Y Zhang, D Remillard, U Onubogu, B Karakyriakou, JN Asiaban, ... Nature Structural & Molecular Biology 30 (8), 1160-1171, 2023 | 6 | 2023 |
| Enabling cancer target validation with genetically encoded systems for ligand-induced protein degradation Y Zhang, MA Erb Current Research in Chemical Biology 1, 100011, 2021 | 6 | 2021 |
| Collateral lethality between HDAC1 and HDAC2 exploits cancer-specific NuRD complex vulnerabilities Y Zhang, D Remillard, U Onubogu, B Karakyriakou, JN Asiaban, ... bioRxiv, 2022 | 4 | 2022 |
| Chemical inhibition of ENL/AF9 YEATS domains in acute leukemia L Garnar-Wortzel, TR Bishop, S Kitamura, N Milosevich, JN Asiaban, ... bioRxiv, 2020.12. 01.406694, 2020 | 2 | 2020 |
| Compounds and methods for treating cancer J Bradner, M Erb, J Qi US Patent 10,464,897, 2019 | 2 | 2019 |
| Inherited blood cancer predisposition through altered transcription elongation J Zhao, LD Cato, UP Arora, EL Bao, SC Bryant, N Williams, Y Jia, ... Cell 187 (3), 642-658. e19, 2024 | 1 | 2024 |
