Microwave-assisted regioselective direct C–H arylation of thiazole derivatives leading to increased σ 1 receptor affinity A Kokornaczyk, D Schepmann, J Yamaguchi, K Itami, B Wünsch MedChemComm 7 (2), 327-331, 2016 | 18 | 2016 |
Synthesis, binding affinity and structure–activity relationships of novel, selective and dual targeting CCR2 and CCR5 receptor antagonists A Junker, AK Kokornaczyk, AJM Zweemer, B Frehland, D Schepmann, ... Organic & Biomolecular Chemistry 13 (8), 2407-2422, 2015 | 18 | 2015 |
Synthesis and biological evaluation of chemokine receptor ligands with 2-benzazepine scaffold S Thum, AK Kokornaczyk, T Seki, M De Maria, NVO Zacarias, H de Vries, ... European Journal of Medicinal Chemistry 135, 401-413, 2017 | 16 | 2017 |
Selective and dual targeting of CCR2 and CCR5 receptors: a current overview A Junker, AK Kokornaczyk, AK Strunz, B Wünsch Chemokines: Chemokines and Their Receptors in Drug Discovery, 187-241, 2015 | 16 | 2015 |
Thiazole‐Based σ1 Receptor Ligands: Diversity by Late‐Stage C−H Arylation of Thiazoles, Structure–Affinity and Selectivity Relationships, and Molecular Interactions AK Kokornaczyk, D Schepmann, J Yamaguchi, K Itami, E Laurini, ... ChemMedChem 12 (13), 1070-1080, 2017 | 7 | 2017 |
Molecular structure of a brominated 2-benzazepinone–a crucial intermediate in the synthesis of novel chemokine CCR2 receptor antagonists AK Kokornaczyk, S Thum, CG Daniliuc, A Junker, B Wünsch Zeitschrift für Naturforschung B 72 (6), 421-424, 2017 | 1 | 2017 |