| Geometrically and conformationally restrained cinnamoyl compounds as inhibitors of HIV-1 integrase: synthesis, biological evaluation, and molecular modeling M Artico, R Di Santo, R Costi, E Novellino, G Greco, S Massa, ... Journal of medicinal chemistry 41 (21), 3948-3960, 1998 | 238 | 1998 |
| Heck reaction on anthraquinone derivatives: ligand, solvent and salt effects W Cabri, I Candiani, S DeBernardinis, F Francalanci, S Penco, R Santo The Journal of Organic Chemistry 56 (20), 5796-5800, 1991 | 222 | 1991 |
| Antimycobacterial pyrroles: synthesis, anti-Mycobacterium tuberculosis activity and QSAR studies R Ragno, GR Marshall, R Di Santo, R Costi, S Massa, R Rompei, M Artico Bioorganic & medicinal chemistry 8 (6), 1423-1432, 2000 | 182 | 2000 |
| 6-[1-(4-Fluorophenyl) methyl-1H-pyrrol-2-yl)]-2, 4-dioxo-5-hexenoic acid ethyl ester a novel diketo acid derivative which selectively inhibits the HIV-1 viral replication in … E Tramontano, F Esposito, R Badas, R Di Santo, R Costi, P La Colla Antiviral research 65 (2), 117-124, 2005 | 145 | 2005 |
| Novel bifunctional quinolonyl diketo acid derivatives as HIV-1 integrase inhibitors: design, synthesis, biological activities, and mechanism of action R Di Santo, R Costi, A Roux, M Artico, A Lavecchia, L Marinelli, ... Journal of medicinal chemistry 49 (6), 1939-1945, 2006 | 122 | 2006 |
| Antifungal Agents. 11. N-Substituted Derivatives of 1-[(Aryl)(4-aryl-1H-pyrrol-3-yl)methyl]-1H-imidazole: Synthesis, Anti-Candida Activity, and QSAR Studies R Di Santo, A Tafi, R Costi, M Botta, M Artico, F Corelli, M Forte, ... Journal of medicinal chemistry 48 (16), 5140-5153, 2005 | 122 | 2005 |
| Natural products as antifungal agents against clinically relevant pathogens R Di Santo Natural product reports 27 (7), 1084-1098, 2010 | 119 | 2010 |
| 2, 6-Bis (3, 4, 5-trihydroxybenzylydene) derivatives of cyclohexanone: novel potent HIV-1 integrase inhibitors that prevent HIV-1 multiplication in cell-based assays R Costi, R Di Santo, M Artico, S Massa, R Ragno, R Loddo, M La Colla, ... Bioorganic & medicinal chemistry 12 (1), 199-215, 2004 | 110 | 2004 |
| Antifungal Agents. 10. New Derivatives of 1-[(Aryl)[4-aryl-1H-pyrrol-3-yl]methyl]-1H-imidazole, Synthesis, Anti-Candida Activity, and Quantitative Structure … A Tafi, R Costi, M Botta, R Di Santo, F Corelli, S Massa, A Ciacci, ... Journal of medicinal chemistry 45 (13), 2720-2732, 2002 | 107 | 2002 |
| Inhibiting the HIV integration process: past, present, and the future R Di Santo Journal of medicinal chemistry 57 (3), 539-566, 2014 | 99 | 2014 |
| Pyrrolnitrin and related pyrroles endowed with antibacterial activities against Mycobacterium tuberculosis R Di Santo, R Costi, M Artico, S Massa, G Lampis, D Deidda, R Pompei Bioorganic & medicinal chemistry letters 8 (20), 2931-2936, 1998 | 91 | 1998 |
| Novel 3, 5-bis (bromohydroxybenzylidene) piperidin-4-ones as coactivator-associated arginine methyltransferase 1 inhibitors: enzyme selectivity and cellular activity D Cheng, S Valente, S Castellano, G Sbardella, R Di Santo, R Costi, ... Journal of medicinal chemistry 54 (13), 4928-4932, 2011 | 89 | 2011 |
| HIV-1 RT-associated RNase H function inhibitors: recent advances in drug development E Tramontano, R Di Santo Current medicinal chemistry 17 (26), 2837-2853, 2010 | 86 | 2010 |
| Structure–activity relationship of pyrrolyl diketo acid derivatives as dual inhibitors of HIV-1 integrase and reverse transcriptase ribonuclease H domain G Cuzzucoli Crucitti, M Métifiot, L Pescatori, A Messore, VN Madia, ... Journal of medicinal chemistry 58 (4), 1915-1928, 2015 | 85 | 2015 |
| Cinnamoyl compounds as simple molecules that inhibit p300 histone acetyltransferase R Costi, R Di Santo, M Artico, G Miele, P Valentini, E Novellino, ... Journal of medicinal chemistry 50 (8), 1973-1977, 2007 | 84 | 2007 |
| Activity of caffeic acid derivatives against Candida albicans biofilm D De Vita, L Friggeri, FD D’Auria, F Pandolfi, F Piccoli, S Panella, ... Bioorganic & medicinal chemistry letters 24 (6), 1502-1505, 2014 | 81 | 2014 |
| Identification of highly conserved residues involved in inhibition of HIV-1 RNase H function by diketo acid derivatives A Corona, FS Di Leva, S Thierry, L Pescatori, G Cuzzucoli Crucitti, ... Antimicrobial agents and chemotherapy 58 (10), 6101-6110, 2014 | 77 | 2014 |
| Design, synthesis and QSAR studies on N-aryl heteroarylisopropanolamines, a new class of non-peptidic HIV-1 protease inhibitors R Di Santo, R Costi, M Artico, S Massa, R Ragno, GR Marshall, P La Colla Bioorganic & medicinal chemistry 10 (8), 2511-2526, 2002 | 72 | 2002 |
| Molecular Modeling of Azole Antifungal Agents Active against Candida albicans. 1. A Comparative Molecular Field Analysis Study A Tafi, J Anastassopoulou, T Theophanides, M Botta, F Corelli, S Massa, ... Journal of medicinal chemistry 39 (6), 1227-1235, 1996 | 70 | 1996 |
| Basic quinolinonyl diketo acid derivatives as inhibitors of HIV integrase and their activity against RNase H function of reverse transcriptase R Costi, M Métifiot, S Chung, G Cuzzucoli Crucitti, K Maddali, L Pescatori, ... Journal of Medicinal Chemistry 57 (8), 3223-3234, 2014 | 66 | 2014 |
