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| Discovery of a potent and selective tyrosine kinase 2 inhibitor: TAK-279 S Leit, J Greenwood, S Carriero, S Mondal, R Abel, M Ashwell, ... Journal of Medicinal Chemistry 66 (15), 10473-10496, 2023 | 7 | 2023 |
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| Allosteric chromenone inhibitors of phosphoinositide 3-kinase (pi3k) for the treatment of disease ED Anderson, SD Aronow, NA Boyles, S Dawadi, ER Hickey, TC Irvin, ... US Patent App. 18/486,620, 2024 | | 2024 |
| Allosteric chromenone inhibitors of phosphoinositide 3-kinase (PI3K) for the treatment of disease ED Anderson, SD Aronow, NA Boyles, X Chen, S Dawadi, ER Hickey, ... US Patent 11,878,970, 2024 | | 2024 |
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| Heterocyclic pericondensed cdc7 kinase inhibitors for the treatment of cancer X Huang, S Mondal, P Ghanakota, N Boyles, L Frye, A Levinson, ... US Patent App. 18/025,465, 2023 | | 2023 |
| Allosteric chromenone inhibitors of phosphoinositide 3-kinase (pi3k) for the treatment of disease ED Anderson, SD Aronow, NA Boyles, MK Dahlgren, F Shulu, ... US Patent App. 18/302,573, 2023 | | 2023 |
| Shape-Based Virtual Screening of a Billion-Compound Library Identifies Mycobacterial Lipoamide Dehydrogenase Inhibitors M Michino, A Beautrait, NA Boyles, A Nadupalli, A Dementiev, S Sun, ... ACS Bio & Med Chem Au 3 (6), 507-515, 2023 | | 2023 |
| 6-heteroaryloxy benzimidazoles and azabenzimidazoles as jak2 inhibitors CE Masse, JR Greenwood, S Mondal, J Xu, P Ghanakota, FM McRobb, ... US Patent App. 18/307,490, 2023 | | 2023 |
| 6-heteroaryloxy benzimidazoles and azabenzimidazoles as JAK2 inhibitors CE Masse, JR Greenwood, S Mondal, J Xu, P Ghanakota, FM McRobb, ... US Patent 11,691,963, 2023 | | 2023 |
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| Discovery of potent, selective, and orally available WEE1 inhibitors that demonstrate increased DNA damage and mitosis in tumor cells leading to tumor regression in vivo S Sun, S Silvergleid, AI Gerasyuto, J Wang, RD Pelletier, A Placzek, ... Cancer Research 82 (12_Supplement), 2570-2570, 2022 | | 2022 |
| Discovery of novel CDC7 inhibitors that disrupt cell cycle dynamics and show anti-proliferative effects in cancer cells L Tsvetkov, A Levinson, X Huang, S Mondal, J Bell, L Tang, R Pelletier, ... Cancer Research 81 (13_Supplement), 1277-1277, 2021 | | 2021 |
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