| Synthesis of a family of spirocyclic scaffolds: building blocks for the exploration of chemical space S Kumar, PD Thornton, TO Painter, P Jain, J Downard, JT Douglas, ... The Journal of organic chemistry 78 (13), 6529-6539, 2013 | 45 | 2013 |
| Design, synthesis, and testing of an 6-O-linked series of benzimidazole based inhibitors of CDK5/p25 P Jain, PT Flaherty, S Yi, I Chopra, G Bleasdell, J Lipay, Y Ferandin, ... Bioorganic & medicinal chemistry 19 (1), 359-373, 2011 | 40 | 2011 |
| Identification of positive allosteric modulators of the D1 dopamine receptor that act at diverse binding sites KD Luderman, JL Conroy, RB Free, N Southall, M Ferrer, M Sanchez-Soto, ... Molecular pharmacology 94 (4), 1197-1209, 2018 | 38 | 2018 |
| Cyclin-dependent kinase 5 (CDK5) controls melanoma cell motility, invasiveness, and metastatic spread—identification of a promising novel therapeutic target S Bisht, J Nolting, U Schütte, J Haarmann, P Jain, D Shah, P Brossart, ... Translational Oncology 8 (4), 295-307, 2015 | 32 | 2015 |
| High-Throughput Screening, Discovery, and Optimization To Develop a Benzofuran Class of Hepatitis C Virus Inhibitors S He, P Jain, B Lin, M Ferrer, Z Hu, N Southall, X Hu, W Zheng, ... ACS combinatorial science 17 (10), 641-652, 2015 | 30 | 2015 |
| Identification of benzimidazole-based inhibitors of the mitogen activated kinase-5 signaling pathway PT Flaherty, I Chopra, P Jain, S Yi, E Allen, J Cavanaugh Bioorganic & medicinal chemistry letters 20 (9), 2892-2896, 2010 | 29 | 2010 |
| Identification of HIV inhibitors guided by free energy perturbation calculations SV Sambasivarao Current Pharmaceutical Design 18 (9), 1199-1216, 2013 | 28 | 2013 |
| Metabolism of JQ1, an inhibitor of bromodomain and extra terminal bromodomain proteins, in human and mouse liver microsomes F Li, KR MacKenzie, P Jain, C Santini, DW Young, MM Matzuk Biology of reproduction 103 (2), 427-436, 2020 | 27 | 2020 |
| Solution-phase synthesis of a diverse library of benzisoxazoles utilizing the [3+ 2] cycloaddition of in situ-generated nitrile oxides and arynes AV Dubrovskiy, P Jain, F Shi, GH Lushington, C Santini, P Porubsky, ... ACS combinatorial science 15 (4), 193-201, 2013 | 25 | 2013 |
| Identification of HIV inhibitors guided by free energy perturbation calculations O Acevedo, Z Ambrose, P T Flaherty, H Aamer, P Jain, S V Sambasivarao Current pharmaceutical design 18 (9), 1199-1216, 2012 | 25 | 2012 |
| Discovery of small molecules targeting the tandem tudor domain of the epigenetic factor UHRF1 using fragment-based ligand discovery L Chang, J Campbell, IO Raji, SKR Guduru, P Kandel, M Nguyen, S Liu, ... Scientific Reports 11 (1), 1121, 2021 | 23 | 2021 |
| Synthesis of Enantiomerically Pure 6-Substituted-Piperazine-2-Acetic Acid Esters as Intermediates for Library Production S Chamakuri, P Jain, SK Reddy Guduru, JW Arney, KR MacKenzie, ... The Journal of organic chemistry 83 (12), 6541-6555, 2018 | 20 | 2018 |
| Steroid receptor coactivator 3 (SRC-3/AIB1) is enriched and functional in mouse and human Tregs BC Nikolai, P Jain, DL Cardenas, B York, Q Feng, NJ McKenna, ... Scientific Reports 11 (1), 3441, 2021 | 14 | 2021 |
| Development of improved SRC-3 inhibitors as breast cancer therapeutic agents L Qin, J Chen, D Lu, P Jain, Y Yu, D Cardenas, X Peng, X Yu, J Xu, ... Endocrine-related cancer 28 (10), 657-670, 2021 | 11 | 2021 |
| Peptidyl Prolyl Isomerase Inhibitors PT Flaherty, P Jain Annual Reports in Medicinal Chemistry 46, 337-349, 2011 | 10 | 2011 |
| Synthesis of Enantiomerically Pure 5-Substituted Piperazine-2-Acetic Acid Esters as Intermediates for Library Production P Jain, IO Raji, S Chamakuri, KR MacKenzie, BT Ebright, C Santini, ... Journal of Organic Chemistry 84 (10), 6040-6064, 2019 | 9 | 2019 |
| Steroid receptor coactivator 3 is a key modulator of regulatory T cell–mediated tumor evasion SJ Han, P Jain, Y Gilad, Y Xia, N Sung, MJ Park, AM Dean, RB Lanz, J Xu, ... Proceedings of the National Academy of Sciences 120 (23), e2221707120, 2023 | 8 | 2023 |
| Suzuki–Miyaura Cross-Coupling of Potassium Organoborates with 6-Sulfonate Benzimidazoles Using Microwave Irradiation P Jain, S Yi, PT Flaherty | 7 | 2013 |
| Structure–activity relationships of benzimidazole-based selective inhibitors of the mitogen activated kinase-5 signaling pathway PT Flaherty, I Chopra, P Jain, D Monlish, J Cavanaugh Bioorganic & medicinal chemistry 18 (22), 8054-8060, 2010 | 7 | 2010 |
| 1-Isopropyl-4-nitro-6-methoxy-1H-benzimidazole MD Moore, P Jain, PT Flaherty, PLD Wildfong Acta Crystallographica Section E: Structure Reports Online 64 (7), o1336-o1337, 2008 | 7 | 2008 |
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