| Design, synthesis and antitumor evaluation of phenyl N-mustard-quinazoline conjugates B Marvania, PC Lee, R Chaniyara, H Dong, S Suman, R Kakadiya, ... Bioorganic & medicinal chemistry 19 (6), 1987-1998, 2011 | 118 | 2011 |
| Potent DNA-directed alkylating agents: Synthesis and biological activity of phenyl N-mustard–quinoline conjugates having a urea or hydrazinecarboxamide linker R Kakadiya, H Dong, A Kumar, D Narsinh, X Zhang, TC Chou, TC Lee, ... Bioorganic & Medicinal Chemistry 18 (6), 2285-2299, 2010 | 72 | 2010 |
| Synthesis and biological activity of stable and potent antitumor agents, aniline nitrogen mustards linked to 9-anilinoacridines via a urea linkage N Kapuriya, K Kapuriya, X Zhang, TC Chou, R Kakadiya, YT Wu, TH Tsai, ... Bioorganic & medicinal chemistry 16 (10), 5413-5423, 2008 | 72 | 2008 |
| Novel Antitumor Indolizino[6,7-b]indoles with Multiple Modes of Action: DNA Cross-Linking and Topoisomerase I and II Inhibition R Chaniyara, S Tala, CW Chen, X Zang, R Kakadiya, LF Lin, CH Chen, ... Journal of medicinal chemistry 56 (4), 1544-1563, 2013 | 70 | 2013 |
| Potent antitumor bifunctional DNA alkylating agents, synthesis and biological activities of 3a-aza-cyclopenta [a] indenes R Kakadiya, H Dong, PC Lee, N Kapuriya, X Zhang, TC Chou, TC Lee, ... Bioorganic & medicinal chemistry 17 (15), 5614-5626, 2009 | 62 | 2009 |
| The development of bis (hydroxymethyl) pyrrole analogs as bifunctional DNA cross-linking agents and their chemotherapeutic potential TL Su, TC Lee, R Kakadiya European Journal of Medicinal Chemistry 69, 609-621, 2013 | 50 | 2013 |
| Combination of bifunctional alkylating agent and arsenic trioxide synergistically suppresses the growth of drug-resistant tumor cells PC Lee, R Kakadiya, TL Su, TC Lee Neoplasia 12 (5), 376-IN2, 2010 | 47 | 2010 |
| Synthesis and antitumor evaluation of novel benzo [d] pyrrolo [2, 1-b] thiazole derivatives R Chaniyara, S Tala, CW Chen, PC Lee, R Kakadiya, H Dong, ... European journal of medicinal chemistry 53, 28-40, 2012 | 42 | 2012 |
| Design, synthesis, and biological evaluation of novel water-soluble N-mustards as potential anticancer agents N Kapuriya, R Kakadiya, H Dong, A Kumar, PC Lee, X Zhang, TC Chou, ... Bioorganic & medicinal chemistry 19 (1), 471-485, 2011 | 41 | 2011 |
| Synthesis and in vitro cytotoxicity of 9-anilinoacridines bearing N-mustard residue on both anilino and acridine rings CH Chen, YW Lin, X Zhang, TC Chou, TJ Tsai, N Kapuriya, R Kakadiya, ... European journal of medicinal chemistry 44 (7), 3056-3059, 2009 | 39 | 2009 |
| Multidrug-resistant cells overexpressing P-glycoprotein are susceptible to DNA crosslinking agents due to attenuated Src/nuclear EGFR cascade-activated DNA repair activity PC Lee, HJ Lee, R Kakadiya, K Sanjiv, TL Su, TC Lee Oncogene 32 (9), 1144-1154, 2013 | 32 | 2013 |
| The novel DNA alkylating agent BO‐1090 suppresses the growth of human oral cavity cancer in xenografted and orthotopic mouse models K Sanjiv, TL Su, S Suman, R Kakadiya, TC Lai, HY Wang, M Hsiao, ... International journal of cancer 130 (6), 1440-1450, 2012 | 30 | 2012 |
| Synthesis of novel imidazo [1, 2-a] pyridine-4-hydroxy-2H-coumarins by Groebke–Blackburn–Bienaymé multicomponent reaction as potential NS5B inhibitors P Manvar, F Shaikh, R Kakadiya, K Mehariya, R Khunt, B Pandey, A Shah Tetrahedron 72 (10), 1293-1300, 2016 | 28 | 2016 |
| Novel bifunctional alkylating agents, 5, 10-dihydropyrrolo [1, 2-b] isoquinoline derivatives, synthesis and biological activity R Chaniyara, N Kapuriya, H Dong, PC Lee, S Suman, B Marvania, ... Bioorganic & medicinal chemistry 19 (1), 275-286, 2011 | 21 | 2011 |
| The synthesis and biological evaluation of new DNA-directed alkylating agents, phenyl N-mustard-4-anilinoquinoline conjugates containing a urea linker B Marvania, R Kakadiya, W Christian, TL Chen, MH Wu, S Suman, K Tala, ... European Journal of Medicinal Chemistry 83, 695-708, 2014 | 19 | 2014 |
| Design and synthesis of 1, 4-dihydropyridine derivatives as anti-cancer agent D Viradiya, S Mirza, F Shaikh, R Kakadiya, A Rathod, N Jain, R Rawal, ... Anti-Cancer Agents in Medicinal Chemistry (Formerly Current Medicinal …, 2017 | 18 | 2017 |
| Inhibition of autophagy enhances DNA damage-induced apoptosis by disrupting CHK1-dependent S phase arrest JS Liou, YC Wu, WY Yen, YS Tang, RB Kakadiya, TL Su, LH Yih Toxicology and applied pharmacology 278 (3), 249-258, 2014 | 17 | 2014 |
| Derivatives of 6-cinnamamido-quinoline-4-carboxamide impair lysosome function and induce apoptosis HH Kuo, R Kakadiya, YC Wu, TL Su, TC Lee, YW Lin, LH Yih Oncotarget 7 (25), 38078, 2016 | 15 | 2016 |
| Fuller’s earth catalyzed rapid synthesis of bis (indolyl) methanes under solvent free condition N Kapuriya, R Kakadiya, MM Savant, AM Pansuriya, CV Bhuva, AS Patel, ... NISCAIR-CSIR, India, 2012 | 12 | 2012 |
| Repairing of N-mustard derivative BO-1055 induced DNA damage requires NER, HR, and MGMT-dependent DNA repair mechanisms CY Kuo, WC Chou, CC Wu, TS Wong, R Kakadiya, TC Lee, TL Su, ... Oncotarget 6 (28), 25770, 2015 | 11 | 2015 |
Dr. Naval P. KapuriyaDepartment of Chemistry and Forensic Science, Bhakta Kavi Narsinh Mehta University, JunagadhVerified email at bknmu.edu.in
