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venkata velvadapu
venkata velvadapu
Scientific Fellow/Director of Chemistry at Senseonics
Verified email at senseonics.com
Title
Cited by
Cited by
Year
Stereochemistry of mephedrone neuropharmacology: enantiomer‐specific behavioural and neurochemical effects in rats
RA Gregg, MH Baumann, JS Partilla, JS Bonano, A Vouga, CS Tallarida, ...
British journal of pharmacology 172 (3), 883-894, 2015
892015
Structure-based design of small-molecule inhibitors of EBNA1 DNA binding blocks Epstein-Barr virus latent infection and tumor growth
TE Messick, GR Smith, SS Soldan, ME McDonnell, JS Deakyne, ...
Science translational medicine 11 (482), eaau5612, 2019
852019
Synthesis of polysubstituted pyrroles from sulfinimines (N-sulfinyl imines)
FA Davis, KA Bowen, H Xu, V Velvadapu
Tetrahedron 64 (19), 4174-4182, 2008
612008
Desmethyl macrolides: synthesis and evaluation of 4, 10-didesmethyl telithromycin
V Velvadapu, I Glassford, M Lee, T Paul, C DeBrosse, D Klepacki, ...
ACS medicinal chemistry letters 3 (3), 211-215, 2012
352012
Total synthesis of (−)-4, 8, 10-tridesmethyl telithromycin
V Velvadapu, T Paul, B Wagh, I Glassford, C DeBrosse, RB Andrade
The Journal of organic chemistry 76 (18), 7516-7527, 2011
342011
Desmethyl macrolides: synthesis and evaluation of 4, 8, 10-tridesmethyl telithromycin
V Velvadapu, T Paul, B Wagh, D Klepacki, O Guvench, A MacKerell Jr, ...
ACS Medicinal Chemistry Letters 2 (1), 68-72, 2011
282011
Concise syntheses of d-desosamine, 2-thiopyrimidinyl desosamine donors, and methyl desosaminide analogues from d-glucose
V Velvadapu, RB Andrade
Carbohydrate research 343 (1), 145-150, 2008
282008
Characterization of a series of 4-aminoquinolines that stimulate caspase-7 mediated cleavage of TDP-43 and inhibit its function
JA Cassel, ME McDonnell, V Velvadapu, V Andrianov, AB Reitz
Biochimie 94 (9), 1974-1981, 2012
272012
Fragment-​based drug discovery
V Velvadapu, BT Farmer, AB Reitz
Practice of Medicinal Chemistry 4, Pages161-180, 2015
242015
Implementation of the CYP Index for the Design of Selective Tryptophan-2, 3-dioxygenase Inhibitors
BT Parr, R Pastor, BD Sellers, Z Pei, FA Jaipuri, GM Castanedo, ...
ACS Medicinal Chemistry Letters 11 (4), 541-549, 2020
222020
Desmethyl macrolides: synthesis and evaluation of 4-desmethyl telithromycin
I Glassford, M Lee, B Wagh, V Velvadapu, T Paul, G Sandelin, ...
ACS Medicinal Chemistry Letters 5 (9), 1021-1026, 2014
212014
Oxidation and reduction potentials of 8-vinyladenosine measured by cyclic voltammetry: Implications for photoinduced electron transfer quenching of a fluorescent adenine analog
M Narayanan, G Kodali, VR Singh, V Velvadapu, RJ Stanley
Journal of Photochemistry and Photobiology A: Chemistry 249, 9-14, 2012
132012
Prodrugs of riluzole and their method of use
GR Smith, AB Reitz, M McDonnell, S Chen, MD Vera, BE Blass, ...
US Patent 9,725,427, 2017
122017
The Practice of Medicinal Chemistry
V Velvadapu, BT Farmer, AB Reitz
ScienceDirect: Amsterdam, Netherlands, 2015
72015
Desmethyl macrolide analogues to address antibiotic resistance: total synthesis and biological evaluation of 4, 8, 10-Tridesmethyl telithromycin
V Velvadapu, T Paul, B Wagh, D Klepacki, O Guvench, A MacKerell Jr, ...
ACS medicinal chemistry letters 2 (1), 68, 2011
72011
TDO2 Inhibitors
X Lin, PW Yuen, R Mendonca, B Parr, R Pastor, Z Pei, L Gazzard, ...
US Patent 10,800,780, 2020
42020
Prodrugs of riluzole and their method of use
GR Smith, AB Reitz, M McDonnell, S Chen, MD Vera, BE Blass, ...
US Patent 10,562,870, 2020
42020
Intramolecular rearrangement of α-amino acid amide derivatives of 2-aminobenzothiazoles
JC Pelletier, V Velvadapu, ME McDonnell, JE Wrobel, AB Reitz
Tetrahedron letters 55 (30), 4193-4195, 2014
32014
Photodesulfinylation of optically active N-sulfinyl amines
FA Davis, T Ramachandar, Y Zhang, J Chai, H Qiu, J Deng, V Velvadapu
Tetrahedron Letters 51 (31), 4042-4044, 2010
32010
Detecting and correcting for changes to an analyte indicator
A DeHennis, M Mortellaro, A Chavan, V Velvadapu, P Huffstetler, THJ Kim, ...
US Patent 10,827,962, 2020
22020
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