| Complex pharmacology of free fatty acid receptors G Milligan, B Shimpukade, T Ulven, BD Hudson Chemical Reviews 117 (1), 67-110, 2017 | 226 | 2017 |
| The pharmacology of TUG-891, a potent and selective agonist of the free fatty acid receptor 4 (FFA4/GPR120), demonstrates both potential opportunity and possible challenges to … BD Hudson, B Shimpukade, AE Mackenzie, AJ Butcher, JD Pediani, ... Molecular pharmacology 84 (5), 710-725, 2013 | 193 | 2013 |
| Discovery of a potent and selective GPR120 agonist B Shimpukade, BD Hudson, CK Hovgaard, G Milligan, T Ulven Journal of medicinal chemistry 55 (9), 4511-4515, 2012 | 189 | 2012 |
| The GPR 120 agonist TUG‐891 promotes metabolic health by stimulating mitochondrial respiration in brown fat M Schilperoort, AD van Dam, G Hoeke, IG Shabalina, A Okolo, ... EMBO molecular medicine 10 (3), e8047, 2018 | 94 | 2018 |
| Non-acidic free fatty acid receptor 4 agonists with antidiabetic activity CMG Azevedo, KR Watterson, ET Wargent, SVF Hansen, BD Hudson, ... Journal of medicinal chemistry 59 (19), 8868-8878, 2016 | 88 | 2016 |
| Selective copper catalysed aromatic N-arylation in water J Engel-Andreasen, B Shimpukade, T Ulven Green chemistry 15 (2), 336-340, 2013 | 76 | 2013 |
| The molecular basis of ligand interaction at free fatty acid receptor 4 (FFA4/GPR120) BD Hudson, B Shimpukade, G Milligan, T Ulven Journal of Biological Chemistry 289 (29), 20345-20358, 2014 | 75 | 2014 |
| Concomitant action of structural elements and receptor phosphorylation determines arrestin-3 interaction with the free fatty acid receptor FFA4 AJ Butcher, BD Hudson, B Shimpukade, E Alvarez-Curto, R Prihandoko, ... Journal of Biological Chemistry 289 (26), 18451-18465, 2014 | 69 | 2014 |
| Novel GPR120 agonist TUG891 modulates fat taste perception and preference and activates tongue-brain-gut axis in mice B Murtaza, A Hichami, AS Khan, B Shimpukade, T Ulven, MH Ozdener, ... Journal of lipid research 61 (2), 133-142, 2020 | 31 | 2020 |
| Treatment with TUG891, a free fatty acid receptor 4 agonist, restores adipose tissue metabolic dysfunction following chronic sleep fragmentation in mice D Gozal, Z Qiao, I Almendros, J Zheng, A Khalyfa, B Shimpukade, T Ulven International Journal of Obesity 40 (7), 1143-1149, 2016 | 31 | 2016 |
| Discovery of a potent free fatty acid 1 receptor agonist with low lipophilicity, low polar surface area, and robust in vivo efficacy SVF Hansen, E Christiansen, C Urban, BD Hudson, CJ Stocker, ... Journal of medicinal chemistry 59 (6), 2841-2846, 2016 | 25 | 2016 |
| Epiminocyclohepta [b] indole analogs as 5-HT6 antagonists AJ Henderson, PR Guzzo, A Ghosh, J Kaur, JM Koo, K Nacro, S Panduga, ... Bioorganic & medicinal chemistry letters 22 (4), 1494-1498, 2012 | 21 | 2012 |
| A concise synthesis of the potent inflammatory mediator 5-oxo-ETE R Tyagi, B Shimpukade, S Blättermann, E Kostenis, T Ulven MedChemComm 3 (2), 195-198, 2012 | 18 | 2012 |
| A newly designed carbohydrate-derived alkylamine promotes Ullmann type C–N coupling catalyzed by copper in water G Zhou, W Chen, S Zhang, X Liu, Z Yang, X Ge, HJ Fan Synlett 30 (02), 193-198, 2019 | 15 | 2019 |
| The pharmacology of a potent and selective agonist, TUG-891, demonstrates both potential opportunity and possible challenges to therapeutic agonism of FFA4 (GPR120) BD Hudson, B Shimpukade, AE Mackenzie, AJ Butcher, JD Pediani, ... Molecular Pharmacology, 2013 | 10 | 2013 |
| An efficient synthesis of (7S, 10R)-2-bromo-5, 6, 7, 8, 9, 10-hexahydro-7, 10-epiminocyclohepta [b] indole: application in the preparation and structural confirmation of a … ML Isherwood, PR Guzzo, AJ Henderson, MM Hsia, J Kaur, K Nacro, ... Tetrahedron: Asymmetry 23 (22-23), 1522-1527, 2012 | 9 | 2012 |
| Process for the preparation of valsartan and its intermediates A Kumar, M Nimbalkar, S Barve, D Metil, R Kelkar, B Shimpukade, ... US Patent App. 11/405,522, 2006 | 7 | 2006 |
| Free fatty acid receptors, FFAR1 and FFAR4, are novel bronchodilator targets in mouse and human precision-cut lung slices J Bourke, R Angeles, C Donovan, M Lam, J Micallef, B Shimpukade, ... European Respiratory Journal 52 (suppl 62), 2018 | 2 | 2018 |
| GPR120 receptor modulators T Ulven, B Shimpukade WO Patent App. 2013/139341A1, 2013 | 1 | 2013 |
| Tetrahydro-benzo [d] azepine derivatives as GPR120 modulators J Brown, S Connolly, SVF Hansen, G MILNE, B SHIMPUKADE, D Smyth, ... US Patent 11,220,483, 2022 | | 2022 |
Graeme MilliganUniversity of GlasgowVerified email at glasgow.ac.uk
