Ewelina Węglarz-Tomczak
Ewelina Węglarz-Tomczak
Postdoc at University of Amsterdam, Swammerdam Institute for Life Sciences
Verified email at uva.nl - Homepage
Title
Cited by
Cited by
Year
Azo dyes—biological activity and synthetic strategy
E Weglarz-Tomczak, L Gorecki
Chemik 66 (12), 1298-1307, 2012
622012
Structure-guided, single-point modifications in the phosphinic dipeptide structure yield highly potent and selective inhibitors of neutral aminopeptidases
S Vassiliou, E Węglarz-Tomczak, Ł Berlicki, M Pawełczak, B Nocek, ...
Journal of medicinal chemistry 57 (19), 8140-8151, 2014
392014
A structural insight into the P1S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective inhibitors of alanine aminopeptidases
E Węglarz-Tomczak, Ł Berlicki, M Pawełczak, B Nocek, A Joachimiak, ...
European journal of medicinal chemistry 117, 187-196, 2016
252016
Identification of methionine aminopeptidase 2 as a molecular target of the organoselenium drug ebselen and its derivatives/analogues: Synthesis, inhibitory activity and …
E Węglarz-Tomczak, M Burda-Grabowska, M Giurg, A Mucha
Bioorganic & medicinal chemistry letters 26 (21), 5254-5259, 2016
212016
Discovery of potent and selective inhibitors of human aminopeptidases ERAP1 and ERAP2 by screening libraries of phosphorus-containing amino acid and dipeptide analogues
E Węglarz-Tomczak, S Vassiliou, A Mucha
Bioorganic & medicinal chemistry letters 26 (16), 4122-4126, 2016
212016
Ebselen as a highly active inhibitor of PLProCoV2
E Weglarz-Tomczak, JM Tomczak, M Talma, S Brul
BioRxiv, 2020
162020
An integrated approach to the ligand binding specificity of Neisseria meningitidis M1 alanine aminopeptidase by fluorogenic substrate profiling, inhibitory studies and …
E Węglarz-Tomczak, M Poręba, A Byzia, Ł Berlicki, B Nocek, R Mulligan, ...
Biochimie 95 (2), 419-428, 2013
162013
An integrated approach to the ligand binding specificity of Neisseria meningitidis M1 alanine aminopeptidase by fluorogenic substrate profiling, inhibitory studies and …
E Węglarz-Tomczak, M Poręba, ...
Biochimie 95 (2), 419-428, 2013
162013
Controlling the Helix Handedness of ααβ‐Peptide Foldamers through Sequence Shifting
M Szefczyk, E Węglarz‐Tomczak, P Fortuna, A Krzysztoń, ...
Angewandte Chemie International Edition 56 (8), 2087-2091, 2017
132017
Discovery of potent inhibitors of PLproCoV2 by screening libraries of selenium-containing compounds
E Weglarz-Tomczak, JM Tomczak, M Giurg, M Burda-Grabowska, S Brul
bioRxiv, 2020
112020
Estimating kinetic constants in the Michaelis–Menten model from one enzymatic assay using Approximate Bayesian Computation
JM Tomczak, E Węglarz‐Tomczak
FEBS letters 593 (19), 2742-2750, 2019
102019
Berlicki Ł., Pawełczak M., Nocek B., Joachimiak A., Mucha A. A structural insight into the P1 S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective …
E Węglarz-Tomczak
Eur. J. Med. Chem 117, 187-196, 2016
82016
Helix-loop-helix peptide foldamers and their use in the construction of hydrolase mimetics
M Drewniak, E Węglarz-Tomczak, K Ożga, E Rudzińska-Szostak, ...
Bioorganic chemistry 81, 356-361, 2018
52018
Berlicki Ł, Pawełczak M, Nocek B, Mulligan R, Joachimiak A, Mucha A. Structure-guided, single-point modifications in the phosphinic dipeptide structure yield highly potent and …
S Vassiliou, E Węglarz-Tomczak
J Med Chem 57, 8140-51, 2014
52014
Berlicki Ł, Nocek B, Mulligan, Joachimiak A, Drąg M, Mucha A. An integrated approach to the ligand binding specificity of Neisseria meningitidis M1 alanine aminopeptidase by …
E Węglarz-Tomczak, M Poręba, A Byzia
Biochimie 95 (2), 419-428, 2013
52013
Identification of ebselen and its analogues as potent covalent inhibitors of papain-like protease from SARS-CoV-2
E Weglarz-Tomczak, JM Tomczak, M Talma, M Burda-Grabowska, ...
Scientific reports 11 (1), 1-10, 2021
42021
Neutral metalloaminopeptidases APN and MetAP2 as newly discovered anticancer molecular targets of actinomycin D and its simple analogs
E Węglarz-Tomczak, M Talma, M Giurg, HV Westerhoff, R Janowsk, ...
Oncotarget 9 (50), 29365-29378, 2018
42018
Enantiomeric α, β-diaminoethylphosphonic acids as potent inhibitors of aminopeptidases—stereoselective synthesis and biological activity
E Węglarz-Tomczak, K Staszewska, M Talma, A Mucha
Tetrahedron Letters 57 (43), 4812-4814, 2016
42016
Differential evolution with reversible linear transformations
JM Tomczak, E Węglarz-Tomczak, AE Eiben
Proceedings of the 2020 Genetic and Evolutionary Computation Conference …, 2020
32020
Barwniki azowe–aktywność biologiczna i strategie syntezy
E Węglarz-Tomczak, Ł Górecki
Chemik 66 (12), 2012
32012
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Articles 1–20