1-(4-Methylphenyl)-2-pyrrolidin-1-yl-pentan-1-one (Pyrovalerone) analogues: a promising class of monoamine uptake inhibitors PC Meltzer, D Butler, JR Deschamps, BK Madras Journal of medicinal chemistry 49 (4), 1420-1432, 2006 | 376 | 2006 |
Further evidence of dopamine transporter dysregulation in ADHD: a controlled PET imaging study using altropane TJ Spencer, J Biederman, BK Madras, DD Dougherty, AA Bonab, E Livni, ... Biological psychiatry 62 (9), 1059-1061, 2007 | 224 | 2007 |
Substituted 3-phenyltropane analogs of cocaine: synthesis, inhibition of binding at cocaine recognition sites, and positron emission tomography imaging PC Meltzer, AY Liang, AL Brownell, DR Elmaleh, BK Madras Journal of medicinal chemistry 36 (7), 855-862, 1993 | 179 | 1993 |
Rapid detection of Parkinson's disease by SPECT with altropane: a selective ligand for dopamine transporters AJ Fischman, AA Bonab, JW Babich, EP Palmer, NM Alpert, DR Elmaleh, ... Synapse 29 (2), 128-141, 1998 | 149 | 1998 |
The discovery of an unusually selective and novel cocaine analog: Difluoropine. Synthesis and inhibition of binding at cocaine recognition sites PC Meltzer, AY Liang, BK Madras Journal of medicinal chemistry 37 (13), 2001-2010, 1994 | 120 | 1994 |
2-Carbomethoxy-3-aryl-8-oxabicyclo [3.2. 1] octanes: potent non-nitrogen inhibitors of monoamine transporters PC Meltzer, AY Liang, P Blundell, MD Gonzalez, Z Chen, C George, ... Journal of medicinal chemistry 40 (17), 2661-2673, 1997 | 106 | 1997 |
A technetium-99m SPECT imaging agent which targets the dopamine transporter in primate brain PC Meltzer, P Blundell, AG Jones, A Mahmood, B Garada, ... Journal of medicinal chemistry 40 (12), 1835-1844, 1997 | 91 | 1997 |
Technepine: A high‐affinity 99mtechnetium probe to label the dopamine transporter in brain by SPECT imaging BK Madras, AG Jones, A Mahmood, RE Zimmerman, B Garada, ... Synapse 22 (3), 239-246, 1996 | 91 | 1996 |
Altropane, a SPECT or PET imaging probe for dopamine neurons: III. Human dopamine transporter in postmortem normal and Parkinson's diseased brain BK Madras, LM Gracz, MA Fahey, D Elmaleh, PC Meltzer, AY Liang, ... Synapse 29 (2), 116-127, 1998 | 78 | 1998 |
2-Carbomethoxy-3-aryl-8-bicyclo [3.2. 1] octanes: potent non-nitrogen inhibitors of monoamine transporters PC Meltzer, P Blundell, YF Yong, Z Chen, C George, MD Gonzalez, ... Journal of medicinal chemistry 43 (16), 2982-2991, 2000 | 73 | 2000 |
Nitrogen‐based drugs are not essential for blockade of monoamine transporters BK Madras, ZB Pristupa, HB Niznik, AY Liang, P Blundell, MD Gonzalez, ... Synapse 24 (4), 340-348, 1996 | 71 | 1996 |
Topical application of spiperone or derivatives thereof for treatment of pathological conditions associated with immune responses RJ Sharpe, KA Arndt, SJ Galli, PC Meltzer, RK Razdan, HP Sard US Patent 5,703,088, 1997 | 61 | 1997 |
Substituted 2-carboxyalkyl-3 (fluorophenyl)-8-(3-halopropen-2-yl) nortropanes and their use as imaging agents for neurodegenerative disorders DR Elmaleh, BK Madras, P Meltzer, RN Hanson US Patent 5,853,696, 1998 | 57 | 1998 |
Altropane, a SPECT or PET imaging probe for dopamine neurons: I. Dopamine transporter binding in primate brain BK Madras, PC Meltzer, AY Liang, DR Elmaleh, J Babich, AJ Fischman Synapse 29 (2), 93-104, 1998 | 57 | 1998 |
Cocaine congeners as PET imaging probes for dopamine terminals AL Brownell, DR Elmaleh, PC Meltzer, TM Shoup, GL Brownell, ... Journal of Nuclear Medicine 37 (7), 1186-1192, 1996 | 57 | 1996 |
Positional Importance of the Nitrogen Atom in Novel Piperidine Analogues of GBR 12909: Affinity and Selectivity for the Dopamine Transporter. AK Dutta, PC Meltzer, BK Madras ChemInform 25 (16), no-no, 1994 | 56 | 1994 |
[11C,127I] Altropane: A highly selective ligand for PET imaging of dopamine transporter sites AJ Fischman, AA Bonab, JW Babich, E Livni, NM Alpert, PC Meltzer, ... Synapse 39 (4), 332-342, 2001 | 54 | 2001 |
2-Carbomethoxy-3-(diarylmethoxy)-1αH,5αH-tropane Analogs: Synthesis and Inhibition of Binding at the Dopamine Transporter and Comparison with … PC Meltzer, AY Liang, BK Madras Journal of medicinal chemistry 39 (2), 371-379, 1996 | 52 | 1996 |
Peptide nucleic acids: synthesis of thymine, adenine, guanine, and cytosine nucleobases PC Meltzer, AY Liang, P Matsudaira The Journal of Organic Chemistry 60 (13), 4305-4308, 1995 | 52 | 1995 |
Altropane, a SPECT or PET imaging probe for dopamine neurons: II. distribution to dopamine‐rich regions of primate brain BK Madras, LM Gracz, PC Meltzer, AY Liang, DR Elmaleh, MJ Kaufman, ... Synapse 29 (2), 105-115, 1998 | 49 | 1998 |